Pipadanu iwuwo Semaglutide CAS 910463-68-2
Apejuwe
Semaglutide (910463-68-2) jẹ oogun egboogi-diabetic ti o ta labẹ awọn orukọ iyasọtọ bii Ozempic, Wegovy, ati Rybelsus.O ti lo lati tọju iru àtọgbẹ 2 ati ṣakoso iwuwo onibaje.Oogun naa n ṣiṣẹ gẹgẹbi glucagon-bi peptide-1 (GLP-1) eniyan nipasẹ jijẹ yomijade hisulini, eyiti o yori si ilọsiwaju iṣelọpọ suga.O ti pin bi abẹrẹ abẹ-ara ti o ni iwọn mita ninu peni ti a kun tẹlẹ, tabi bi fọọmu ẹnu.Ọkan ninu awọn anfani rẹ lori awọn oogun antidiabetic miiran ni pe o ni akoko pipẹ ti iṣe, nitorinaa, abẹrẹ lẹẹkan ni ọsẹ kan to.
Nlo
A lo Semaglutide lati ṣakoso iru àtọgbẹ 2 pẹlu awọn ayipada igbesi aye, gẹgẹbi awọn ihamọ ijẹẹmu ati iṣẹ ṣiṣe ti ara pọ si.O tun ṣiṣẹ nipa fifalẹ gbigbe ounjẹ nipasẹ ikun ati pe o le dinku ifẹkufẹ ati fa pipadanu iwuwo.Ko si awọn ijabọ ti a tẹjade ti hepatotoxicity ti a sọ si itọju ailera semaglutide.
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Mechanism ti igbese
Semaglutide jẹ agonist olugba olugba glucagon-bi peptide-1.O mu iṣelọpọ insulin pọ si, homonu ti o dinku ipele suga ẹjẹ.O tun han lati mu idagbasoke ti awọn sẹẹli β wa ninu oronro, eyiti o jẹ aaye ti iṣelọpọ insulin.O tun ṣe idiwọ glucagon, eyiti o jẹ homonu ti o mu suga ẹjẹ pọ si.Ni afikun, o dinku gbigbe ounjẹ nipasẹ jijẹ jijẹ ati fa fifalẹ tito nkan lẹsẹsẹ ninu ikun.Ni ọna yii o dinku ọra ara.
Ti ibi aṣayan iṣẹ-ṣiṣe
Semaglutide (Rybelsus, Ozempic, NN9535, OG217SC, NNC 0113-0217), afọwọṣe glucagon-like peptide 1 (GLP-1), jẹ agonist olugba GLP-1 pẹlu agbara fun itọju iru 2 diabetes mellitus. (T2DM).
Iṣakojọpọ & Ifijiṣẹ
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