SARM SR9011 Pharmaceutical Raw Powder Mo Faʻateleina le Faʻamalositino Tumau CAS 1379686-30-2
SR9011 Fa'amatalaga vave
Cas Numera 1379686-29-9
Synonyms 3-(((4-chlorobenzyl)((5-nitrothiophen-2-yl)methyl)amino)methyl)-N-pentylpyrrolidine-
1-carboxamide
Fuafua C23H31ClN4O3S
Molucelar mamafa 479.03524
SR9011Fa'amatalaga
O le SR9011 o se monomer methacrylate fa'apitoa e maua ai le pipii fa'apitoa i u'amea
mea'ai.
SR9011 ua fautuaina mo le faʻaaogaina i faʻamaʻi faʻamalolo faʻamalolo, faʻamaufaʻailoga, ma plastisols faʻavae PVC.
Fa'aaoga tulaga o le 5% i le 10% i le mamafa e fautuaina.
O le SR9011 o se REV-ERB malosi ma fa'apitoa.E lelei fo'i i vivo plasma/fai'ai fa'aalia.
O le faʻaogaina faaniukilia REV-ERB-α ma REV-ERB-β o loʻo i ai se sao taua i le faʻatonutonuina o faʻamatalaga.
o polotini autu o le uati, ave le pao i gaioiga ma metabolism.Pulega o le SR9011 suia
amio circadian ma le mamanu circadian o le fa'aaliga autu o le uati i le hypothalami o isumu.
O le fa'ata'ita'iga fa'asologa o le fa'asologa o kenera metabolic i le ate, musele skeletal ma
ua toe suia foi aano o le tino, ma i'u ai i le faateleina o tupe faaalu.Togafitiga o mea taumafa
isumu lapo'a ma le SR9011 fa'aitiitia le puta e ala i le fa'aitiitia o le ga'o ma fa'aleleia lelei le dyslipidemia ma le hyperglycaemia.O nei fa'ai'uga o lo'o fa'ailoa mai ai le fa'aogaina ole REV-ERB ligand e fa'atatau ile vaila'au
e mafai ona aoga le pa'u o le circadian i le togafitia o faaletonu o le moe faapea foi ma gasegase metabolic.
![SR9009 (2)](http://www.chem-peptide-steroids.com/uploads/SR9009-2-300x295.png)
![SR9009](http://www.chem-peptide-steroids.com/uploads/SR9009-300x298.png)
![SR9009 (1)](http://www.chem-peptide-steroids.com/uploads/SR9009-1.png)
Fa'afefea ona fa'aoga SR9011?
In vitro: SR9011 na faʻaaogaina i le 5-10 μM faʻatonuga i vitro ma i suʻega feaveaʻi.
In vivo: IP pulega o le SR9011 na faʻaaogaina i le 100 mg / kg tasi pe faalua i le aso mo le 12-30
aso i fa'ata'ita'iga isumu eseese.
Fa'asologa o le SR9009 ma le SR9011
Aitema | Fa'amatalaga | I'uga |
Fa'aaliga | O se pauta e leai se manogi, toetoe lava pa'epa'e pe pa'epa'e | pasi |
Fa'ailoaga | Ole taimi ole taofi ole tumutumu tele ole fa'amaonia i le RS | pasi |
Ma'imau ile Fa'amago | E le sili atu i le 0.5% | 0.33% |
Su'ega(HPLC) | Le itiiti ifo i le 99.0% | 99.59% |
Toega mumu | E le sili atu i le 0.1% | pasi |
Uamea mamafa | Le sili atu i le 20 ppm | pasi |
afifiina & Tiliva
![包装运输](http://www.chem-peptide-steroids.com/uploads/包装运输2-300x300.jpg)
![包装](http://www.chem-peptide-steroids.com/uploads/包装1-300x245.png)
![2CF15DBA-28DD-4a76-8CFE-0A38764249E5](http://www.chem-peptide-steroids.com/uploads/2CF15DBA-28DD-4a76-8CFE-0A38764249E5.png)