Kurwanya Estrogene Nolvadex (Citrate ya Tamoxifen) Ifu yubaka umubiri kuri PCT CAS 10540-29-1
Citrate ya Tamoxifen (Nolvadex) Ibisobanuro
Irindi zina: Nolvadex
CAS: 10540-29-1
MF: C32H37NO8
MW: 563.64
Kugaragara: ifu yera-yera-ifu
Imikoreshereze: estrogene antagonist, antineoplastique
Ikoreshwa: Gukoresha mukuvura kanseri yamabere yateye imbere, kanseri yintanga nayo irakora, kandi ibisubizo byiza hamwe nibindi biyobyabwenge birwanya kanseri
Gupakira: Nkibisabwa abakiriya
Ijambo ryibanze: Citrate ya Tamoxifen, uruganda rwa citrate ya Tamoxifen
Citrate ya Tamoxifen (Nolvadex) COA
| Ibizamini | Ibisobanuro | Ibisubizo by'ibizamini |
| Ibisobanuro | Ifu ya kirisiti yera | Ifu ya kirisiti yera |
| Kumenyekanisha | IR, UV ihuza | Hindura |
| Gutakaza kumisha | .5 0.5ml | 0.21ml |
| Ibisigisigi byo gutwikwa | Ntabwo arenze 0.2% | 0.06ml |
| Icyuma | Ntabwo arenze 0.005% | 0.0018% |
| Ibyuma biremereye | Ntabwo arenze 0.001% | 0.0006% |
| Ibintu bifitanye isano | Igiteranyo: Ntabwo arenze 1.0% Umuntu ku giti cye: Ntabwo arenze 0.5% | 0.32% 0.14% |
| E-isomer | Ntabwo arenze 0.3% | 0.19% |
| Umwanda uhindagurika | Guhuza | Guhuza |
| Suzuma | 99.0 ~ 101.0% | 99.51% |
| Umwanzuro | Ihuze na USP30 | |
Citro ya Tamoxifen (Nolvadex) Ibisobanuro
Nolvadex ni icyamamare kandi gifite imbaraga zo guhitamo Estrogen Receptor Modulator (SERM) bakunze kwita anti-estrogene.Ariko, nubwo kuba antagonist nayo ni agonist kuko mubyukuri izakora nka estrogene mubice bimwe na bimwe byumubiri mugihe ikora nka anti-estrogene mubindi bice.Nka imwe muri SERM ya kera cyane ku isoko ikomeje gukoreshwa mubuvuzi, mugihe Nolvadex nayo ikoreshwa nabakoresha anabolike steroid ntabwo ari anabolicsteroid.Iyi ni ingingo y'ingenzi kuko bamwe bakunze kwitiranywa nikoreshwa ryayo muri steroid.Nolvadex ni SERM gusa.
Nolvadex, izwi ku izina rya Tamoxifen Citrate, yakozwe bwa mbere mu 1961 na ICI ubu AstraZeneca ku izina ry'ubucuruzi Nolvadex.SERM yakozwe mu kuvura kanseri y'ibere, cyane cyane kanseri y'ibere yitabira imisemburo.Icyakora, yakoreshejwe kandi mu gukumira kanseri y'ibere.Noneho dufite abakoresha anabolic steroid, kandi byavumbuwe kera ko Nolvadex yari ifite umwanya mubantu nkabo.Nolva, nkuko bisanzwe bizwi, irashobora gukoreshwa nka anti-estrogene mugihe cya anabolike steroid cycle kugirango wirinde ingaruka ziterwa na estrogene.Irakoreshwa kandi mubice bigize gahunda yo gukira ya Post Cycle Therapy (PCT), niyo ngingo isanzwe kandi yingirakamaro yo gukoresha kubakoresha steroid.
Gupakira & Gutanga
